Trenbolone Acetate Injection

(Intramuscular Injection 100mg/1ml)

Composition

Each 1 ml. of Trenbolone Acetate contains 100 mg. in Oily base. Ethyl oleate quantity sufficient and Benzyl alcohol.

Pharmacodynamics

Trenbolone Acetate is anabolic steroid having binding affinity for the androgen receptor. When administered by intramuscular injection, it is metabolized and increases nitrogen uptake by muscles, leading to an increase in the rate of protein synthesis. Trenbolone is an highly effective anabolic steroid, promoting protein synthesis, as well as creating a positive nitrogen balance. It is an appetite stimulant and improves the conversion of protein. Trenbolone Acetate has a secondary effect on appetite stimulation, thus reducing the amount of adipose tissue being deposited in the body, and decreasing the rate of catabolism.

Pharmacokinetic

Trenbolone Acetate is an anabolic steroid contains steroid ester. The half -life of a steroid ester is mostly dependent on its ratio of fat solubility to water solubility; the longer chain the ester, the higher this ratio, and thus the longer the half-life. Trenbolone Acetate has a half-life 5-7 days with 100% bioavailability on intramuscular administration. Trenbolone is not metabolised by aromatase or 5a-reductase into estrogenic compounds such as estradiol, or into DHT, thus it does not cause any water retention which is normally associated with highly androgenic steroidal methandrostenolone . When metabolised it get excreted in urine as conjugates that can be hydrolyzed with beta- glucuronidase. This implies that trenbolone leaves the body as beta-glucuronides or sulfates, which means mostly non metabolized.

Indications and Usage

On administration of Trenbolone Acetate there is an increase in muscle hardness, muscular strength. In combination with a protein rich diet, Trenbolone Acetate speeds up the metabolism and accelerates the burning of adipose tissue. The high androgenic effect prevents a possible muscle- break down syndrome and accelerates the regeneration of muscles tissue.

Dosage and Administration

A normal dosage can range from 100 mg/week up to 229.5 mg/week. Due to short metabolic half-life of Trenbolone Acetate it can be taken twice or thrice a week. Effective Dose (Men): 100 mg -229.5 mg/week. Effective Dose (Women): Not established. Active life: 5-7 days.

Side effects

Side effects includes nausea, vomiting, insomnia, poor sleep patterns, high blood pressure and increased aggression, increased libido, severe sweating during the nighttime. Acne and hair loss only occur rarely which might be due to the fact that the substance is not converted into dihydrotestosterone (DHT), when administered more than 100 mg per week, reports nausea, headaches, and loss of appetite.

Contraindications

Trenbolone Acetate contraindicated in kidney dysfunction, hypertension, cardiac patients. Also it is contraindicated in infants, pregnancy and nursing mothers. Trenbolone Acetate should not be used in patients with known hypersensitivity to drug or any of it's

Warning & Precautions

When administered parenterally, there is tightness in the chest, and a metallic taste in the back of the mouth, followed by an uncontrollable violent cough & bronchoconstriction. Trenbolone reduces endogenous T3 thyroid levels and increases prolactin levels. Thus to overcome the unwanted side effects that could be caused by rise in prolactin levels, 25 mcg T3 should be used throughout a trenbolone treatment. When administered in high dosages over several weeks, the patient often reports unusually dark colored urine. In extreme cases blood can be excreted through the urine, as clear sign of kidney damage. It is therefore essential that during Trenbolone Acetate therapy, the patient should increase the daily fluid consumption to help flush the kidneys Trenbolone Acetate should not be given to females, as it causes virilization even in small doses. The side effect noted in are: acne, androgenically caused hair loss on the scalp, irregular menstrual cycles, missed periods, much higher libido, aggressiveness, deep voice, clitoral hypertrophy, and increased hair growth on face and on the legs. The last three side effects are mostly irreversible changes.

Storage

Store in cool dry place below 30°C, Protect from light. Keep out of reach of children.

Presentation

10 ml. vial is packed in a carton tray. Each carton tray includes 10 ml. vial and information leaflet.